Browsing by Contributors Cosconati, Sandro

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PreviewIssue DateTitleContributor(s)
2018 JMC Volume 61 Issue 13 July (20).pdf.jpg20184-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX InhibitorsSalerno, Silvia; Barresi, Elisabetta; Amendola, Giorgio; Berrino, Emanuela; Milite, Ciro; Marini, Anna Maria; Settimo, Federico Da; Novellino, Ettore; Supuran, Claudiu T; Cosconati, Sandro; Taliani, Sabrina
2012medicine article a (127).pdf.jpg2012Adenosine Receptor AntagonistsTaliani, Sabrina; Pugliesi, Isabella; Barresi, Elisabetta; Simorini, Francesca; Salerno, Silvia; Motta, Concettina La; Marini, Anna Maria; Cosimelli, Barbara; Cosconati, Sandro; Maro, Salvatore Di; Marinelli, Luciana; Daniele, Simona; Trincavelli, Maria Letizia; Greco, Giovanni; Novellino, Ettore; Martini, Claudia; Settimo, Federico Da; Farmaceutiche, Scienze; Pisa, Universita; Bonanno, Via; Farmaceutica, Chimica; Federico, Napoli; Montesano, Via D
2014medicine article a (245).pdf.jpg2014Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptaseCosti, Roberta; Métifiot, Mathieu; Chung, Suhman; Cuzzucoli Crucitti, Giuliana; Maddali, Kasthuraiah; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Scipione, Luigi; Tortorella, Silvano; Di Leva, Francesco Saverio; Cosconati, Sandro; Mari
2012medicine article a (785).pdf.jpg2012Benzofuroxane Derivatives as Multi-E ff ective Agents for the Treatment of Cardiovascular Diabetic Complications. Synthesis, Functional Evaluation, and Molecular Modeling StudiesSartini, Stefania; Cosconati, Sandro; Marinelli, Luciana; Barresi, Elisabetta; Maro, Salvatore Di; Simorini, Francesca; Taliani, Sabrina; Salerno, Silvia; Marini, Anna Maria; Settimo, Federico Da; Novellino, Ettore; Motta, Concettina La; Farmacia, Dipartimento; Pisa, Universita; Bonanno, Via
2015 JMC Volume 58 Issue 20 October (3).pdf.jpg2015Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic ActivityEadsforth, Thomas C.; Pinto, Andrea; Luciani, Rosaria; Tamborini, Lucia; Cullia, Gregorio; De Micheli, Carlo; Marinelli, Luciana; Cosconati, Sandro; Novellino, Ettore; Lo Presti, Leonardo; Cordeiro Da Silva, Anabela; Conti, Paola; Hunter, William N.; Costi, Maria P.
2017 JMC Volume 60 Issue 19 October (13).pdf.jpg2017Computer-Aided Identi fi cation and Lead Optimization of Dual Murine Double Minute 2 and 4 Binders: Structure − Activity Relationship Studies and Pharmacological ActivityGiustiniano, Mariateresa; Daniele, Simona; Pelliccia, Sveva; Pietra, Valeria La; Pietrobono, Deborah; Brancaccio, Diego; Cosconati, Sandro; Messere, Anna; Giuntini, Stefano; Cerofolini, Linda; Fragai, Marco; Luchinat, Claudio; Taliani, Sabrina; Regina, Giuseppe La; Set
2015 JMC Volume 58 Issue 15 August (28).pdf.jpg2015Deepening the Topology of the Translocator Protein Binding Site by Novel N,N-Dialkyl-2-arylindol-3-ylglyoxylamidesBarresi, Elisabetta; Bruno, Agostino; Taliani, Sabrina; Cosconati, Sandro; Da Pozzo, Eleonora; Salerno, Silvia; Simorini, Francesca; Daniele, Simona; Giacomelli, Chiara; Marini, Anna Maria; La Motta, Concettina; Marinelli, Luciana; Cosimelli, Barbara; Novellino, Ettor
2011medicine article a (74).pdf.jpg2011Design , Synthesis , and Functionalization of Dimeric Peptides Targeting Chemokine Receptor CXCR4Demmer, Oliver; Dijkgraaf, Ingrid; Schumacher, Udo; Marinelli, Luciana; Cosconati, Sandro; Gourni, Eleni; Kessler, Horst
2015 JMC Volume 58 Issue 7 April (6).pdf.jpg2015Design, Synthesis, and Biological Evaluation of Novel 2-((2-(4-(Substituted)phenylpiperazin-1-yl)ethyl)amino)-5′- <i>N</i> -ethylcarboxamidoadenosines as Potent and Selective Agonists of the A <sub>2A</sub> Adenosine ReceptorPreti, Delia; Baraldi, Pier Giovanni; Saponaro, Giulia; Romagnoli, Romeo; Aghazadeh Tabrizi, Mojgan; Baraldi, Stefania; Cosconati, Sandro; Bruno, Agostino; Novellino, Ettore; Vincenzi, Fabrizio; Ravani, Annalisa; Borea, Pier Andrea; Varani, Katia
2017 JMchemistry Volume 60 Issue 16 August (10).pdf.jpg2017Development of Novel Peptide Based Michael Acceptors Targeting Rhodesain and Falcipain ‑ 2 for the Treatment of Neglected Tropical Diseases (NTDs)Previti, Santo; Ettari, Roberta; Cosconati, Sandro; Amendola, Giorgio; Chouchene, Khawla; Wagner, Annika; Hellmich, Ute A; Ulrich, Kathrin; Krauth-siegel, R Luise; Wich, Peter R; Schmid, Ira; Schirmeister, Tanja; Gut, Jiri; Rosenthal, Philip J; Grasso, Silvana; Zappala, Maria
2019 JournalofMedicalChemistry Volume 62 Issue 5 March (30).pdf.jpg2019Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1/2 (GLP/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal StructureMilite, Ciro; Feoli, Alessandra; Horton, John R; Rescigno, Donatella; Cipriano, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Pepe, Giacomo; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Cheng, Xiaodong; Castellano, Sabrina; Sbardella, Gianluca
2017 JMchemistry Volume 60 Issue 17 September (15).pdf.jpg2017Dual MET and SMO Negative Modulators Overcome Resistance to EGFR Inhibitors in Human Nonsmall Cell Lung CancerMorgillo, Floriana; Amendola, Giorgio; Maria, Carminia; Corte, Della; Giacomelli, Chiara; Botta, Lorenzo; Maro, Salvatore Di; Messere, Anna; Ciaramella, Vincenza; Taliani, Sabrina; Marinelli, Luciana; Trincavelli, Maria Letizia; Martini, Claudia; Novellino, Ettore; Ciardiello, Fortunato; Cosconati, Sandro
2017 JMchemistry Volume 60 Issue 18 September (19).pdf.jpg2017Exploiting the 4 ‑ Phenylquinazoline Sca ff old for the Development of High A ffi nity Fluorescent Probes for the Translocator Protein (TSPO)Milite, Ciro; Barresi, Elisabetta; Pozzo, Eleonora Da; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Δ Gianluca; Settimo, Federico Da; Novellino, Ettore; Cosconati, Sandro; Castellano, Δ Sabrina; Taliani, Sabrina; Martini, Claudia; Farmacia, Dipartimento; Pisa, Universita; Bonanno, Via
2013medicine article a (778).pdf.jpg2013Exploring the Chemical Space of G ‑ Quadruplex Binders: Discovery of a Novel Chemotype Targeting the Human Telomeric SequenceSaverio, Francesco; Leva, Di; Zizza, Pasquale; Cingolani, Chiara; Angelo, Carmen D; Pagano, Bruno; Amato, Jussara; Salvati, Erica; Sissi, Claudia; Pinato, Odra; Marinelli, Luciana; Cavalli, Andrea; Cosconati, Sandro; Novellino, Ettore; Randazzo, Antonio; Biroccio, Annam
2017 JMC Volume 60 Issue 9 May (2).pdf.jpg2017Lead Discovery of Dual G Quadruplex Stabilizers and Poly(ADP ribose) Polymerases (PARPs) Inhibitors: A New Avenue in Anticancer TreatmentSalvati, Erica; Botta, Lorenzo; Amato, Jussara; Di Leva, Francesco Saverio; Zizza, Pasquale; Gioiello, Antimo; Pagano, Bruno; Graziani, Grazia; Tarsounas, Madalena; Randazzo, Antonio; Novellino, Ettore; Biroccio, Annamaria; Cosconati, Sandro
2016 JMC Volume 59 Issue 10 May (8).pdf.jpg2016Lead Optimization of 2 ‑ Phenylindolylglyoxylyldipeptide Murine Double Minute (MDM)2/Translocator Protein (TSPO) Dual Inhibitors for the Treatment of GliomasDaniele, Simona; Pietra, Valeria La; Barresi, Elisabetta; Maro, Salvatore Di; Pozzo, Eleonora Da; Robello, Marco; Motta, Concettina La; Cosconati, Sandro; Taliani, Sabrina; Marinelli, Luciana; Novellino, Ettore; Martini, Claudia; Settimo, Federico Da
2013medicine article a (322).pdf.jpg2013Ligand Based Approach to L ‑ Type Calcium Channel by Imidazo[2,1 ‑ b ]thiazole-1,4-Dihydropyridines: from Heart Activity to Brain A ffi nityLocatelli, Alessandra; Cosconati, Sandro; Micucci, Matteo; Leoni, Alberto; Marinelli, Luciana; Bedini, Andrea; Ioan, Pierfranco; Spampinato, Santi Mario; Novellino, Ettore; Chiarini, Alberto; Budriesi, Roberta
2016 JMC Volume 59 Issue 12 June (23).pdf.jpg2016Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of GlaucomaVullo, Daniela; Durante, Mariaconcetta; Saverio, Francesco; Leva, Di; Cosconati, Sandro; Masini, Emanuela; Scozzafava, Andrea; Novellino, Ettore; Supuran, Claudiu T; Carta, Fabrizio; Scienti, Polo; Bioinorganica, Chimica; Lastruccia, Via; Fiorentino, Sesto
2015 JMC Volume 58 Issue 11 June (7).pdf.jpg2015N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse TranscriptasePescatori, Luca; M??tifiot, Mathieu; Chung, Suhman; Masoaka, Takashi; Cuzzucoli Crucitti, Giuliana; Messore, Antonella; Pupo, Giovanni; Madia, Valentina Noemi; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Di Leva, Francesco Saverio; Cosconati, Sandro
2011medicine article a (290).pdf.jpg2011New 2-Heterocyclyl-imidazo [ 2 , 1- i ] purin-5-one Derivatives as Potent and Selective Human A 3 Adenosine Receptor AntagonistsBaraldi, Pier Giovanni; Preti, Delia; Zaid, Abdel Naser; Saponaro, Giulia; Tabrizi, Mojgan Aghazadeh; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Allan R; Varani, Katia; Cosconati, Sandro; Maro, Salvatore Di; Marinelli, Luciana; Novellino, Ettore; Borea, Pier Andrea